PMID

Data

Article Title

Organization

Ion channels as therapeutic targets: a drug discovery perspective.

Pfizer

Selective influence on contextual memory: physiochemical properties associated with selectivity of benzodiazepine ligands at GABAA receptors containing the alpha5 subunit.

Moltech

Exploring subtype selectivity and metabolic stability of a novel series of ligands for the benzodiazepine binding site of the GABAA receptor.

Novartis Institutes For Biomedical Research

Tricyclic pyridones as functionally selective human GABAA alpha 2/3 receptor-ion channel ligands.

The Neuroscience Research Centre

Synthesis and biological evaluation of 7,8,9,10-tetrahydroimidazo[1,2-c]pyrido[3,4-e]pyrimdin-5(6H)-ones as functionally selective ligands of the benzodiazepine receptor site on the GABA(A) receptor.

Neurogen

The amylase inhibitor montbretin A reveals a new glycosidase inhibition motif.

University Of British Columbia

Structure-guided design of a high affinity inhibitor to human CtBP.

University Of Massachusetts Medical School