PMID

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Structure-activity relationship studies on 1-(2-oxopropyl)indole-5-carboxylic acids acting as inhibitors of cytosolic phospholipase A

University Of M£Nster

Design, synthesis, and biological evaluation of 3-(1-Aryl-1H-indol-5-yl)propanoic acids as new indole-based cytosolic phospholipase A2a inhibitors.

Asubio Pharma

Inhibition of group IVA cytosolic phospholipase A2 by thiazolyl ketones in vitro, ex vivo, and in vivo.

University Of Athens

1-(5-Carboxyindol-1-yl)propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha: synthesis and properties of bioisosteric benzimidazole, benzotriazole and indazole analogues.

University Of M£Nster

1-(2-Carboxyindol-5-yloxy)propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha: synthesis, biological activity, metabolic stability, and solubility.

University Of M£Nster

1-Indol-1-yl-propan-2-ones and related heterocyclic compounds as dual inhibitors of cytosolic phospholipase A(2)alpha and fatty acid amide hydrolase.

University Of M£Nster

Reactions of functionalized sulfonamides: application to lowering the lipophilicity of cytosolic phospholipase A2alpha inhibitors.

Wyeth Research

 

Dicarboxylic acid inhibitors of phospholipase A₂

TBA

Inhibitory effect of synthetic C-C biflavones on various phospholipase A(2)s activity.

Yeungnam University

1-(5-Carboxy- and 5-carbamoylindol-1-yl)propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha: bioisosteric replacement of the carboxylic acid and carboxamide moiety.

University Of MüNster

Discovery of Ecopladib, an indole inhibitor of cytosolic phospholipase A2alpha.

Wyeth Research

Design and synthesis of 1-indol-1-yl-propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha.

University Of MüNster

1,2,4-Oxadiazolidin-3,5-diones and 1,3,5-triazin-2,4,6-triones as cytosolic phospholipase A2alpha inhibitors.

Wyeth Research

Inhibition of cytosolic phospholipase A2alpha: hit to lead optimization.

Wyeth Research

Structure-activity relationships of indole cytosolic phospholipase A(2)alpha inhibitors: substrate mimetics.

Wyeth Research

Pyrrolidine inhibitors of human cytosolic phospholipase A(2).

Shionogi

Substrate-Specific Inhibition Constants for Phospholipase A

University Of California

?-Lactones: A Novel Class of Ca

National And Kapodistrian University Of Athens

Synthesis and characterization of 3-arylquinazolinone and 3-arylquinazolinethione derivatives as selective estrogen receptor beta modulators.

Bristol-Myers Squibb

Discovery and evaluation of 3-(5-thien-3-ylpyridin-3-yl)-1H-indoles as a novel class of KDR kinase inhibitors.

Merck Research Laboratories