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18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Optimization of furin inhibitors to protect against the activation of influenza hemagglutinin H5 and Shiga toxin.EBI
Universit£
Design, synthesis, and structure-activity relationship studies of a potent PACE4 inhibitor.EBI
Universit£
The Multi-Leu peptide inhibitor discriminates between PACE4 and furin and exhibits antiproliferative effects on prostate cancer cells.EBI
Universit£
Furin inhibitors: importance of the positive formal charge and beyond.EBI
Torrey Pines Institute For Molecular Studies
New substrate analogue furin inhibitors derived from 4-amidinobenzylamide.EBI
Philipps University Marburg
New furin inhibitors based on weakly basic amidinohydrazones.EBI
Philipps University Marburg
Synthesis and optimization of thiadiazole derivatives as a novel class of substrate competitive c-Jun N-terminal kinase inhibitors.EBI
Institute For Medical Research
Potent inhibitors of furin and furin-like proprotein convertases containing decarboxylated P1 arginine mimetics.EBI
Philipps University Marburg
Discovery of 2-(5-nitrothiazol-2-ylthio)benzo[d]thiazoles as novel c-Jun N-terminal kinase inhibitors.EBI
Institute For Medical Research
Modeling the activity of furin inhibitors using artificial neural network.EBI
Mahidol University
Targeting host cell furin proprotein convertases as a therapeutic strategy against bacterial toxins and viral pathogens.EBI
Institute For Medical Research
Notch Antagonists: Potential Modulators of Cancer and Inflammatory Diseases.EBI
Centre Hospitalier Universitaire Vaudois (Chuv)
Synthesis of tight binding inhibitors and their action on the proprotein-processing enzyme furin.EBI
Friedrich Miescher-Institut
Improving the Selectivity of PACE4 Inhibitors through Modifications of the P1 Residue.EBI
TBA
Increasing C-Terminal Hydrophobicity Improves the Cell Permeability and Antiproliferative Activity of PACE4 Inhibitors against Prostate Cancer Cell Lines.EBI
Universit£
Positional Scanning Identifies the Molecular Determinants of a High Affinity Multi-Leucine Inhibitor for Furin and PACE4.EBI
University Of Gdansk
Discovery of novel secretory phospholipase A2 inhibitors using virtual screen.BDB
Peking University