PMID

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Article Title

Organization

Synthesis and Evaluation of Novel Tetrahydronaphthyridine CXCR4 Antagonists with Improved Drug-like Profiles.

Emory University

Structure-Based Design and Optimization of FPPQ, a Dual-Acting 5-HT

Jagiellonian University Medical College

Discovery, Structure-Activity Relationships, and In Vivo Evaluation of Novel Aryl Amides as Brain Penetrant Adaptor Protein 2-Associated Kinase 1 (AAK1) Inhibitors for the Treatment of Neuropathic Pain.

Bristol Myers Squibb

Structure activity relationship of 3-nitro-2-(trifluoromethyl)-2H-chromene derivatives as P2Y

National Institute Of Diabetes And Digestive And Kidney Diseases

Structure-Activity Relationship of Heterocyclic P2Y

National Institute Of Diabetes And Digestive And Kidney Diseases

Discovery, structure-activity relationship study and biological evaluation of 2-thioureidothiophene-3-carboxylates as a novel class of C-X-C chemokine receptor 2 (CXCR2) antagonists.

University Of Michigan

Synthesis and pharmacological evaluation of piperidine (piperazine)-amide substituted derivatives as multi-target antipsychotics.

Jiangsu Ocean University

Small Molecules Selectively Targeting Sigma-1 Receptor for the Treatment of Neurological Diseases.

Soochow University

Ifenprodil Stereoisomers: Synthesis, Absolute Configuration, and Correlation with Biological Activity.

Westf£Lische Wilhelms-Universit£T M£Nster

Leveraging an Open Science Drug Discovery Model to Develop CNS-Penetrant ALK2 Inhibitors for the Treatment of Diffuse Intrinsic Pontine Glioma.

Ontario Institute For Cancer Research

Exploration of Alternative Scaffolds for P2Y

National Institute Of Diabetes And Digestive And Kidney Diseases

Isolation and Synthesis of Veranamine, an Antidepressant Lead from the Marine Sponge

University Of Mississippi

Structure-Based Design of 3-(4-Aryl-1H-1,2,3-triazol-1-yl)-Biphenyl Derivatives as P2Y14 Receptor Antagonists.

National Institute Of Diabetes And Digestive And Kidney Diseases

Synthesis of spiro-2,6-dioxopiperazine and spiro-2,6-dioxopyrazine scaffolds using amino acids in a three-component reaction to generate potential Sigma-1 (?

Memorial Sloan Kettering Cancer Center

Discovery, Optimization, and Characterization of ML417: A Novel and Highly Selective D

National Institute Of Neurological Disorders And Stroke

Leveraging a Low-Affinity Diazaspiro Orthosteric Fragment to Reduce Dopamine D

University Of Pennsylvania

Defining Structure-Functional Selectivity Relationships (SFSR) for a Class of Non-Catechol Dopamine D

University Of North Carolina At Chapel Hill

Investigation of the Adrenergic and Opioid Binding Affinities, Metabolic Stability, Plasma Protein Binding Properties, and Functional Effects of Selected Indole-Based Kratom Alkaloids.

University Of Florida

Design and in Vivo Characterization of A

Medical College Of Wisconsin

Functionalized 6-(Piperidin-1-yl)-8,9-Diphenyl Purines as Peripherally Restricted Inverse Agonists of the CB1 Receptor.

Rti International

Bicyclic ?-Iminophosphonates as High Affinity Imidazoline I

University Of Barcelona

Benzyl Phenylsemicarbazides: A Chemistry-Driven Approach Leading to G Protein-Biased Dopamine D

Friedrich-Alexander-Universit£T Erlangen-N£Rnberg

3-Amino-chromanes and Tetrahydroquinolines as Selective 5-HT

University Of Minnesota Twin Cities

A SARS-CoV-2 protein interaction map reveals targets for drug repurposing.

Qbi Covid-19 Research Group (Qcrg)