19 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
Data
Article Title
Organization
Novel biguanide-based derivatives scouted as TAAR1 agonists: Synthesis, biological evaluation, ADME prediction and molecular docking studies.
University of Genoa
Discovery and Characterization of 2-Aminooxazolines as Highly Potent, Selective, and Orally Active TAAR1 Agonists.
Roche Innovation Center Basel
Optimisation of imidazole compounds as selective TAAR1 agonists: discovery of RO5073012.
F. Hoffmann-La Roche
Trace amine-associated receptor 1 is a stereoselective binding site for compounds in the amphetamine class.
Research Triangle Institute
Selective antagonists of mouse trace amine-associated receptor 1 (mTAAR1): discovery of EPPTB (RO5212773).
F. Hoffmann-La Roche
Amiodarone and its putative metabolites fail to activate wild type hTAAR1.
Rti International
Structure-activity correlations for beta-phenethylamines at human trace amine receptor 1.
Rti International
Progress in mechanistically novel treatments for schizophrenia.
Novartis Institutes For Biomedical Research
Rational design, chemical synthesis and biological evaluation of novel biguanides exploring species-specificity responsiveness of TAAR1 agonists.
University of Genoa
