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35 articles for L De Petrocellis


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Cmpds
Data
Article Title
Organization
15
Neuroactive and Anti-inflammatory Frankincense Cembranes: A Structure-Activity Study.EBI
University of Eastern Piedmont
36
Arylboronic acids as dual-action FAAH and TRPV1 ligands.EBI
Sapienza University of Rome
21
TRPA1 channels as targets for resveratrol and related stilbenoids.EBI
Sapienza University of Rome
6
Discovery of non-electrophilic capsaicinoid-type TRPA1 ligands.EBI
University of Eastern Piedmont
54
Structure-activity relationships of the prototypical TRPM8 agonist icilin.EBI
National Research Council
35
Structure-affinity relationships and pharmacological characterization of new alkyl-resorcinol cannabinoid receptor ligands: Identification of a dual cannabinoid receptor/TRPA1 channel agonist.EBI
University of Siena
39
Effect of acyclic monoterpene alcohols and their derivatives on TRP channels.EBI
Sapienza University of Rome
18
3-Ylidenephthalides as a new class of transient receptor potential channel TRPA1 and TRPM8 modulators.EBI
Sapienza University of Rome
33
Biaryl tetrazolyl ureas as inhibitors of endocannabinoid metabolism: modulation at the N-portion and distal phenyl ring.EBI
Sapienza University of Rome
25
Tetrahydro-ß-carboline derivatives targeting fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channels.EBI
Sapienza University of Rome
35
Modulation of thermo-transient receptor potential (thermo-TRP) channels by thymol-based compounds.EBI
Sapienza University of Rome
10
Structure-activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): The side chain benzylic methylene.EBI
University of Eastern Piedmont
19
New tetrazole-based selective anandamide uptake inhibitors.EBI
Sapienza University of Rome
13
Structure-activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): the homovanillyl moiety.EBI
University of Eastern Piedmont
22
Synthesis and biological evaluation of [6]-gingerol analogues as transient receptor potential channel TRPV1 and TRPA1 modulators.EBI
Sapienza University of Rome
3
Bioactive prenylogous cannabinoid from fiber hemp (Cannabis sativa).EBI
Universita` Del Piemonte Orientale
22
(-)-Menthylamine derivatives as potent and selective antagonists of transient receptor potential melastatin type-8 (TRPM8) channels.EBI
Sapienza University of Rome
25
Synthesis and biological evaluation of piperazinyl carbamates and ureas as fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channel dual ligands.EBI
Sapienza University of Rome
3
Taste-guided identification of high potency TRPA1 agonists from Perilla frutescens.EBI
Università
12
Phytochemical Characterization and TRPA1/TRPM8 Modulation Profile of the Cannabigerol-Rich EBI
University of Naples Federico Ii
31
-Guided Rational Drug Design and Synthesis of Novel 4-(Thiophen-2-yl)butanamides as Potent and Selective TRPV1 Agonists.EBI
Magna Gracia University
11
Oxyhomologues of anandamide and related endolipids: chemoselective synthesis and biological activity.EBI
University of Piemonte Orientale
22
The taming of capsaicin. Reversal of the vanilloid activity of N-acylvanillamines by aromatic iodination.EBI
University of Piemonte Orientale
3
Discovery of a Remarkable Methyl Shift Effect in the Vanilloid Activity of Triterpene Amides.EBI
National Research Council (Icb-Cnr)
2
Cannabitwinol, a Dimeric Phytocannabinoid from Hemp, EBI
University of Naples Federico Ii
28
Synthetic bioactive olivetol-related amides: The influence of the phenolic group in cannabinoid receptor activity.EBI
University of Siena
39
Tetrahydroisoquinoline-Derived Urea and 2,5-Diketopiperazine Derivatives as Selective Antagonists of the Transient Receptor Potential Melastatin 8 (TRPM8) Channel Receptor and Antiprostate Cancer Agents.EBI
National Research Council
28
N-Acylvanillamides: development of an expeditious synthesis and discovery of new acyl templates for powerful activation of the vanilloid receptor.EBI
Istituto Per La Chimica Di Molecole Di Interesse Biologico
51
Elongation of the Hydrophobic Chain as a Molecular Switch: Discovery of Capsaicin Derivatives and Endogenous Lipids as Potent Transient Receptor Potential Vanilloid Channel 2 Antagonists.EBI
National Research Council (Cnr)
6
Iodine-mediated cyclization of cannabigerol (CBG) expands the cannabinoid biological and chemical space.EBI
University of Naples Federico II
2
Iodine-Promoted Aromatization of p-Menthane-Type Phytocannabinoids.EBI
University of Eastern Piedmont
16
JAK kinase inhibitor compounds for treatment of respiratory diseaseBDB
Theravance Biopharma R&D Ip
19
Identification and Biological Evaluation of a Series of 1H-Benzo[de]isoquinoline-1,3(2H)-diones as Hepatitis C Virus NS5B Polymerase Inhibitors.BDB
Irbm, Mrl Rome
17
P1' oxadiazole protease inhibitors with excellent activity against native and protease inhibitor-resistant HIV-1.BDB
Merck Research Laboratories