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32 articles for A Agarwal


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Three-dimensional quantitative structure-activity relationships of 5-HT receptor binding data for tetrahydropyridinylindole derivatives: a comparison of the Hansch and CoMFA methods.EBI
University of Georgia
N-fused imidazoles as novel anticancer agents that inhibit catalytic activity of topoisomerase IIa and induce apoptosis in G1/S phase.EBI
National Institute of Pharmaceutical Education and Research (NIPER)
N-(1,3-Diaryl-3-oxopropyl)amides as a new template for xanthine oxidase inhibitors.EBI
Indo-Soviet Friendship College of Pharmacy
A rational approach for the design and synthesis of 1-acetyl-3,5-diaryl-4,5-dihydro(1H)pyrazoles as a new class of potential non-purine xanthine oxidase inhibitors.EBI
Indo-Soviet Friendship College of Pharmacy
Is structural hybridization invoking new dimensions for antimalarial drug discovery research?EBI
University of Delhi
Structure-activity relationship of 6-methylidene penems bearing 6,5 bicyclic heterocycles as broad-spectrum beta-lactamase inhibitors: evidence for 1,4-thiazepine intermediates with C7 R stereochemistry by computational methods.EBI
Wyeth Research
Discovery of proline sulfonamides as potent and selective hepatitis C virus NS5b polymerase inhibitors. Evidence for a new NS5b polymerase binding site.EBI
Wyeth Research
Development of BRD4 inhibitors as anti-inflammatory agents and antidotes for arsenicals.EBI
Southern Research
Structure-activity relationship of 6-methylidene penems bearing tricyclic heterocycles as broad-spectrum beta-lactamase inhibitors: crystallographic structures show unexpected binding of 1,4-thiazepine intermediates.EBI
Wyeth Research
Tetrazole derivatives as TRPA1 inhibitorsBDB
Boehringer Ingelheim International
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASEBDB
Vertex Pharmaceuticals
TYK2 inhibitors and uses thereofBDB
Nimbus Lakshmi
Isoquinoline derivatives and use thereofBDB
Purdue Pharma
Haloallylamine indole and azaindole derivative inhibitors of lysyl oxidases and uses thereofBDB
Pharmaxis
Selective inhibitors of protein arginine methlytransferase 5 (PRMT5)BDB
Prelude Therapeutics
Indole Chloropyridinyl Ester-Derived SARS-CoV-2 3CLpro Inhibitors: Enzyme Inhibition, Antiviral Efficacy, Structure-Activity Relationship, and X-ray Structural Studies.BDB
Purdue University
Potent and selective inhibitors of monoamine transporters; method of making; and use thereofBDB
The United States of America, As Represented By The Secretary, Department of Health and Human Services
1-pyrazolyl-3-(4-((2-anilinopyrimidin-4-yl) oxy) napththalen-1-yl) ureas as P38 MAP knase inhibitorsBDB
Respivert
Heterocyclic inhibitors of ATR kinaseBDB
University Of Texas
Pyrimido-pyridazinone compounds and methods of use thereofBDB
Asan Biosciences
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitorsBDB
Eli Lilly
Thieno- and furo[2,3-d]pyrimidine-2,4[1H,3H]-dione derivativesBDB
Hydra Biosciences
Inhibition of the alpha- and beta-carbonic anhydrases from the gastric pathogen Helycobacter pylori with anions.BDB
Universit�� Degli Studi Di Firenze
17a-hydroxylase/C17,20-lyase inhibitorsBDB
Novartis
Substituted cycloocta[5,6]pyrido[4,3,2-de]phthalazines as PARP inhibitorsBDB
Beigene
Mechanism of Flavoprotein l-6-Hydroxynicotine Oxidase: pH and Solvent Isotope Effects and Identification of Key Active Site Residues.BDB
University of Texas Health Science Center
Nitrogen-containing saturated heterocyclic compoundBDB
Mitsubishi Tanabe Pharma
Methods for increasing the stabilization of hypoxia inducible factor-αBDB
Aerpio Therapeutics
Molecular Mechanism for Isoform-Selective Inhibition of Acyl Protein Thioesterases 1 and 2 (APT1 and APT2).BDB
University of Michigan
The A128T resistance mutation reveals aberrant protein multimerization as the primary mechanism of action of allosteric HIV-1 integrase inhibitors.BDB
The Ohio State University
Inhibitors of sodium glucose cotransporter 1BDB
Lexicon Pharmaceuticals
4-arylazo-3,5-diamino-1H-pyrazole CDK inhibitors: SAR study, crystal structure in complex with CDK2, selectivity, and cellular effects.BDB
Palacky University