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21 articles for LY Hu


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Design, synthesis, and pharmacological evaluation of conformationally constrained analogues of N,N'-diaryl- and N-aryl-N-aralkylguanidines as potent inhibitors of neuronal Na+ channels.EBI
Cambridge Neuroscience
Synthesis and pharmacological evaluation of N-(2,5-disubstituted phenyl)-N'-(3-substituted phenyl)-N'-methylguanidines as N-methyl-D-aspartate receptor ion-channel blockers.EBI
Cambridge Neuroscience
Pantolactams as androgen receptor antagonists for the topical suppression of sebum production.EBI
Pfizer
Rational design of a topical androgen receptor antagonist for the suppression of sebum production with properties suitable for follicular delivery.EBI
Pfizer
 
Synthesis and characterization of N-(acenaphth-5-yl)-N'-(4-methoxynaphth-1-yl)guanidine as a glutamate release inhibitor and potential anti-ischemic agentEBI
TBA
Diphenyl ethers as androgen receptor antagonists for the topical suppression of sebum production.EBI
Pfizer
4-(Alkylthio)- and 4-(arylthio)-benzonitrile derivatives as androgen receptor antagonists for the topical suppression of sebum production.EBI
Pfizer
Virtual screening for Raf-1 kinase inhibitors based on pharmacophore model of substituted ureas.EBI
China Pharmaceutical University
(1R,2S)-4-(2-cyano-cyclohexyl-oxy)-2-trifluoromethyl-benzonitrile, a potent androgen receptor antagonist for stimulating hair growth and reducing sebum production.EBI
Pfizer
Synthesis and biological evaluation of amino-pyridines as androgen receptor antagonists for stimulating hair growth and reducing sebum production.EBI
Pfizer
Preparation of 4-aryl-2-trifluoromethylbenzonitrile derivatives as androgen receptor antagonists for topical suppression of sebum production.EBI
Pfizer
The design and synthesis of human branched-chain amino acid aminotransferase inhibitors for treatment of neurodegenerative diseases.EBI
Pfizer
Synthesis of a series of 4-benzyloxyaniline analogues as neuronal N-type calcium channel blockers with improved anticonvulsant and analgesic properties.EBI
Warner-Lambert
Structure-activity relationship at the proximal phenyl group in a series of non-peptidyl N-type calcium channel antagonists.EBI
Parke-Davis Pharmaceutical Research
Structure-activity relationship of N-methyl-N-aralkyl-peptidylamines as novel N-type calcium channel blockers.EBI
Warner-Lambert
Multiple parallel synthesis of N,N-dialkyldipeptidylamines as N-type calcium channel blockers.EBI
Warner-Lambert
Synthesis and biological evaluation of substituted 4-(OBz)phenylalanine derivatives as novel N-type calcium channel blockers.EBI
Warner-Lambert
N,N-dialkyl-dipeptidylamines as novel N-type calcium channel blockers.EBI
Warner-Lambert
Synthesis and structure-activity studies of N,N'-diarylguanidine derivatives. N-(1-naphthyl)-N'-(3-ethylphenyl)-N'-methylguanidine: a new, selective noncompetitive NMDA receptor antagonist.EBI
Cambridge Neuroscience
Aryl- and heteroarylcarbonyl derivatives of hexahydroindenopyridine and octahydrobenzoquinolineBDB
Vitae Pharmaceuticals
Small-molecule HSP90 inhibitorsBDB
Memorial Sloan-Kettering Cancer Center