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21 articles for SA Boyd


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
C5-Alkyl-2-methylurea-Substituted Pyridines as a New Class of Glucokinase Activators.EBI
Amgen
Discovery of 2-pyridylureas as glucokinase activators.EBI
Array Biopharma
Discovery of 6-[5-(4-fluorophenyl)-3-methyl-pyrazol-4-yl]-benzoxazin-3-one derivatives as novel selective nonsteroidal mineralocorticoid receptor antagonists.EBI
Takeda Pharmaceutical
Identification of a new class of glucokinase activators through structure-based design.EBI
Array Biopharma
Design, synthesis, and structure-activity relationships of dihydrofuran-2-one and dihydropyrrol-2-one derivatives as novel benzoxazin-3-one-based mineralocorticoid receptor antagonists.EBI
Takeda Pharmaceutical
 
Synthesis and In Vitro evaluation of fused ring heterocyle-containing angiotensin II antagonists.EBI
TBA
Non-charged thiamine analogs as inhibitors of enzyme transketolase.EBI
Array Biopharma
Synthesis, in vitro and in vivo activity of thiamine antagonist transketolase inhibitors.EBI
Array Biopharma
2-(Alkylamino)nicotinic acid and analogs. Potent angiotensin II antagonists.EBI
Abbott Laboratories
Identification of benzoxazin-3-one derivatives as novel, potent, and selective nonsteroidal mineralocorticoid receptor antagonists.EBI
Takeda Pharmaceutical
Novel acyl coenzyme A (CoA): diacylglycerol acyltransferase-1 inhibitors: synthesis and biological activities of diacylethylenediamine derivatives.EBI
Takeda Pharmaceutical
Prodrug thiamine analogs as inhibitors of the enzyme transketolase.EBI
Array Biopharma
Selective inhibition of ICAM-1 and E-selectin expression in human endothelial cells. 2. Aryl modifications of 4-(aryloxy)thieno[2,3-c]pyridines with fine-tuning at C-2 carbamides.EBI
Abbott Laboratories
Discovery of inhibitors of cell adhesion molecule expression in human endothelial cells. 1. Selective inhibition of ICAM-1 and E-selectin expression.EBI
Abbott Laboratories
Discovery and preclinical development of AR453588 as an anti-diabetic glucokinase activator.EBI
Array Biopharma
Novel Series of Potent Glucokinase Activators Leading to the Discovery of AM-2394.EBI
Amgen
Pyrrolidine-3-carboxylic acids as endothelin antagonists. 3. Discovery of a potent, 2-nonaryl, highly selective ETA antagonist (A-216546).EBI
Abbott Laboratories
2,4-Diarylpyrrolidine-3-carboxylic acids--potent ETA selective endothelin receptor antagonists. 1. Discovery of A-127722.EBI
Abbott Laboratories
Nonpeptide renin inhibitors with good intraduodenal bioavailability and efficacy in dog.EBI
Abbott Laboratories
C-terminal modifications of nonpeptide renin inhibitors: improved oral bioavailability via modification of physicochemical properties.EBI
Abbott Laboratories
DELIVERY OF THERAPEUTIC ALKALOID COMPOUNDSBDB
Sensorium Therapeutics