BindingDB

The first public molecular recognition database, BindingDB supports research, education and practice in drug discovery, pharmacology and related fields.

BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.5M data for 737K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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29 articles for G Appendino

The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Neuroactive and Anti-inflammatory Frankincense Cembranes: A Structure-Activity Study.EBI
University of Eastern Piedmont
Turmeric Sesquiterpenoids: Expeditious Resolution, Comparative Bioactivity, and a New Bicyclic Turmeronoid.EBI
University of Eastern Piedmont
Discovery of non-electrophilic capsaicinoid-type TRPA1 ligands.EBI
University of Eastern Piedmont
STAT-3 inhibitory bisabolanes from Carthamus glaucus.EBI
University of Naples Federico II
Structure-activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): The side chain benzylic methylene.EBI
University of Eastern Piedmont
Modulation of the transient receptor potential vanilloid channel TRPV4 by 4alpha-phorbol esters: a structure-activity study.EBI
Ku Leuven
Synthesis and biological evaluation of hyperforin analogues. Part I. Modification of the enolized cyclohexanedione moiety.EBI
University of Milan
Structure-activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): the homovanillyl moiety.EBI
University of Eastern Piedmont
Synthesis and evaluation of phorboid 20-homovanillates: discovery of a class of ligands binding to the vanilloid (capsaicin) receptor with different degrees of cooperativity.EBI
Institute
Bioactive prenylogous cannabinoid from fiber hemp (Cannabis sativa).EBI
Universita` Del Piemonte Orientale
Oxyhomologues of anandamide and related endolipids: chemoselective synthesis and biological activity.EBI
University of Piemonte Orientale
The taming of capsaicin. Reversal of the vanilloid activity of N-acylvanillamines by aromatic iodination.EBI
University of Piemonte Orientale
ΔEBI
Eth Z�Rich
Homologues and isomers of noladin ether, a putative novel endocannabinoid: interaction with rat cannabinoid CB(1) receptors.EBI
Discaff
Discovery of a Remarkable Methyl Shift Effect in the Vanilloid Activity of Triterpene Amides.EBI
National Research Council (Icb-Cnr)
Cannabitwinol, a Dimeric Phytocannabinoid from Hemp, EBI
University of Naples Federico Ii
The Oxidation of Phytocannabinoids to Cannabinoquinoids.EBI
University of Eastern Piedmont
Triterpenoid Hydroxamates as HIF Prolyl Hydrolase Inhibitors.EBI
University of Eastern Piedmont
Identification of a Strigoterpenoid with Dual Nrf2 and Nf-κB Modulatory Activity.EBI
University of Eastern Piedmont
Dissecting the pharmacophore of curcumin. Which structural element is critical for which action?EBI
University of Eastern Piedmont
Vanilloid receptor TRPV1 antagonists as the next generation of painkillers. Are we putting the cart before the horse?EBI
Hospital of The University of Pennsylvania
N-Acylvanillamides: development of an expeditious synthesis and discovery of new acyl templates for powerful activation of the vanilloid receptor.EBI
Istituto Per La Chimica Di Molecole Di Interesse Biologico
Iodine-mediated cyclization of cannabigerol (CBG) expands the cannabinoid biological and chemical space.EBI
University of Naples Federico II
Electrophilic Triterpenoid Enones: A Comparative Thiol-Trapping and Bioactivity Study.EBI
University of Eastern Piedmont
Iodine-Promoted Aromatization of p-Menthane-Type Phytocannabinoids.EBI
University of Eastern Piedmont
The Bibenzyl Canniprene Inhibits the Production of Pro-Inflammatory Eicosanoids and Selectively Accumulates in Some Cannabis sativa Strains.EBI
University of Eastern Piedmont
JAK kinase inhibitor compounds for treatment of respiratory diseaseBDB
Theravance Biopharma R&D Ip