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21 articles for TA Branchek


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of alpha 1a-adrenergic receptor antagonists based on the L-type Ca2+ channel antagonist niguldipine.EBI
Synaptic Pharmaceutical
Substituted furo[3,2-b]pyridines: novel bioisosteres of 5-HT 1F receptor agonists.EBI
Eli Lilly
Novel potent 5-HT(1F) receptor agonists: structure-activity studies of a series of substituted N-[3-(1-methyl-4-piperidinyl)-1H-pyrrolo[3,2-b]pyridin-5-yl]amides.EBI
Eli Lilly
Design and synthesis of novel alpha1a adrenoceptor-selective dihydropyridine antagonists for the treatment of benign prostatic hyperplasia.EBI
Synaptic Pharmaceutical
Design, synthesis and evaluation of substituted triarylnipecotic acid derivatives as GABA uptake inhibitors: identification of a ligand with moderate affinity and selectivity for the cloned human GABA transporter GAT-3.EBI
Synaptic Pharmaceutical
2-amino-2-oxazolines as subtype selective alpha(2) adrenoceptor agonists.EBI
Lundbeck Research Usa
Identification of a dihydropyridine as a potent alpha1a adrenoceptor-selective antagonist that inhibits phenylephrine-induced contraction of the human prostate.EBI
New York University Medical Center
Carboxamide derivatives and use thereofBDB
Purdue Pharma
2,5-disubstituted-pyridyl nicotinic ligands, and methods of use thereofBDB
Georgetown University
5,5-bicyclic oxazole orexin receptor antagonistsBDB
Merck Sharp & Dohme
Compounds and compositions for inhibiting the activity of SHP2BDB
Novartis
1-sulfonyl piperidine derivatives as modulators of prokineticin receptorsBDB
Takeda Pharmaceutical
Compounds and methods for kinase modulation, and indications thereforBDB
Plexxikon
2-(1H-indazol-3-yl)-3H-imidazo[4,5-B]pyridine and therapeutic uses thereofBDB
Samumed
Pyrazines as modulators of GPR6BDB
Takeda Pharmaceutical
Substituted 6,5-fused bicyclic heteroaryl compoundsBDB
Epizyme
Identification of a potent new chemotype for the selective inhibition of PDE4.BDB
Nih
Specific Targeting of Highly Conserved Residues in the HIV-1 Reverse Transcriptase Primer Grip Region. 2. Stereoselective Interaction to Overcome the Effects of Drug Resistant Mutations.BDB
Universita Di Siena
Carbonic anhydrase inhibitors: the membrane-associated isoform XV is highly inhibited by inorganic anions.BDB
Universita Degli Studi Di Firenze
Novel inhibitors of fatty acid amide hydrolase.BDB
Bristol-Myers Squibb
Novel mechanistic class of fatty acid amide hydrolase inhibitors with remarkable selectivity.BDB
Pfizer