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17 articles for DR Sibley


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Novel Analogues of (R)-5-(Methylamino)-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one (Sumanirole) Provide Clues to Dopamine D2/D3 Receptor Agonist Selectivity.EBI
Columbia University College of Physicians and Surgeons
Discovery, optimization, and characterization of novel D2 dopamine receptor selective antagonists.EBI
National Center For Advancing Translational Sciences
N-(3-fluoro-4-(4-(2-methoxy or 2,3-dichlorophenyl)piperazine-1-yl)butyl)arylcarboxamides as selective dopamine D3 receptor ligands: critical role of the carboxamide linker for D3 receptor selectivity.EBI
National Institute On Drug Abuse-Intramural Research Program
Pharmacology and Therapeutic Potential of Benzothiazole Analogues for Cocaine Use Disorder.EBI
High Point University
Development of pyrimidone D1 dopamine receptor positive allosteric modulators.EBI
National Institutes of Health
Discovery, Optimization, and Characterization of ML417: A Novel and Highly Selective DEBI
National Institute of Neurological Disorders and Stroke
Dopamine DEBI
Rowan University
Synthesis and Pharmacological Characterization of Novel trans-Cyclopropylmethyl-Linked Bivalent Ligands That Exhibit Selectivity and Allosteric Pharmacology at the Dopamine DEBI
National Institute On Drug Abuse
Method of treatment with histamine-3 receptor inverse agonistBDB
Suven Life Sciences
Specific inhibitors of cytochrome P450 26 retinoic acid hydroxylaseBDB
University of Washington Through Its Center For Commercialization
Substituted nicotinimide inhibitors of BTK and their preparation and use in the treatment of cancer, inflammation and autoimmune diseaseBDB
Guangzhou Innocare Pharma Tech
Benzimidazol-2-amines as MIDH1 inhibitorsBDB
Bayer Pharma Aktiengesellschaft
Serine/threonine kinase inhibitorsBDB
Genentech
Anchored plasticity opens doors for selective inhibitor design in nitric oxide synthase.BDB
The Scripps Research Institute
Rhodanine derivatives as selective protease inhibitors against bacterial toxins.BDB
Burnham Institute For Medical Research
Alpha,Beta-cyclic-beta-benzamido hydroxamic acids: Novel oxaspiro[4.4]nonane templates for the discovery of potent, selective, orally bioavailable inhibitors of tumor necrosis factor-alpha converting enzyme (TACE).BDB
Bristol-Myers Squibb