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30 articles for P Delagrange


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
New quinolinic derivatives as melatonergic ligands: Synthesis and pharmacological evaluation.EBI
Universities of Lille
Melatonergic ligands: Design, synthesis and pharmacological evaluation of novel series of naphthofuranic derivatives.EBI
University of Lille
Synthesis of 2-arylfuro[3,2-b]pyridines: Effect of the C2-aryl group on melatoninergic activity.EBI
Orleans University
Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1-Benzyl-2-acylaminomethyl-tetrahydroquinolines.EBI
University of Urbino
Synthesis of new N-(arylcyclopropyl)acetamides and N-(arylvinyl)acetamides as conformationally-restricted ligands for melatonin receptors.EBI
Paris-Sud University
Novel and selective partial agonists of 5-HT3 receptors. 2. Synthesis and biological evaluation of piperazinopyridopyrrolopyrazines, piperazinopyrroloquinoxalines, and piperazinopyridopyrroloquinoxalines.EBI
University of Caen Normandy
Novel selective and partial agonists of 5-HT3 receptors. Part 1. Synthesis and biological evaluation of piperazinopyrrolothienopyrazines.EBI
University of Caen Normandy
First tricyclic oximino derivatives as 5-HT3 ligands.EBI
University of Caen Normandy
Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT(1) melatoninergic ligands.EBI
University of Lille
Design, synthesis and pharmacological evaluation of new series of naphthalenic analogues as melatoninergic (MT1/MT2) and serotoninergic 5-HT2C dual ligands (I).EBI
University of Lille
Design and synthesis of 2-phenylimidazo[1,2-a]pyridines as a novel class of melatonin receptor ligands.EBI
Orleans University
Preparation and pharmacological evaluation of a novel series of 2-(phenylthio)benzo[b]thiophenes as selective MT2 receptor ligands.EBI
University of Lille
Design and synthesis of naphthalenic derivatives as new ligands at the melatonin binding site MT3.EBI
University of Lille
Design and synthesis of 1-(2-alkanamidoethyl)-6-methoxy-7-azaindole derivatives as potent melatonin agonists.EBI
Orleans University
Synthesis of 3-phenylnaphthalenic derivatives as new selective MT(2) melatoninergic ligands.EBI
University of Lille 2
Design and synthesis of benzofuranic derivatives as new ligands at the melatonin-binding site MT3.EBI
Université
3-[5-(4,5-dihydro-1H-imidazol-2-yl)-furan-2-yl]phenylamine (Amifuraline), a promising reversible and selective peripheral MAO-A inhibitor.EBI
Università
Design and synthesis of naphthalenic dimers as selective MT1 melatoninergic ligands.EBI
Université
Synthesis and structure-affinity-activity relationships of novel benzofuran derivatives as MT(2) melatonin receptor selective ligands.EBI
Institut De Chimie Pharmaceutique Albert Lespagnol
Synthesis of nitroindole derivatives with high affinity and selectivity for melatoninergic binding sites MT(3).EBI
Institut De Chimie Pharmaceutique Albert Lespagnol
Quinazoline and phthalazine derivatives as novel melatonin receptor ligands analogues of agomelatine.EBI
Umr-S1172 - Jparc - Centre De Recherche Jean-Pierre Aubert Neurosciences Et Cancer
Synthesis of phenalene and acenaphthene derivatives as new conformationally restricted ligands for melatonin receptors.EBI
Paris-Sud University
Original Design of Fluorescent Ligands by Fusing BODIPY and Melatonin Neurohormone.EBI
Orleans University
Melatonergic properties of the (+)- and (-)-enantiomers of N-(4-methoxy-2,3-dihydro-1H-phenalen-2-yl)amide derivatives.EBI
University of Paris
Synthesis of 2-amido-2,3-dihydro-1H-phenalene derivatives as new conformationally restricted ligands for melatonin receptors.EBI
Cnrs-Biocis
Design and synthesis of new naphthalenic derivatives as ligands for 2-[125I]iodomelatonin binding sites.EBI
Cnrs-Biocis
Synthesis and structure-activity relationships of novel naphthalenic and bioisosteric related amidic derivatives as melatonin receptor ligands.EBI
Institut De Chimie Pharmaceutique
Synthesis and biological evaluation of new naphtho- and quinolinocyclopentane derivatives as potent melatoninergic (MTEBI
Univ. Lille
Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands.EBI
University of Parma
Synthesis and SAR of piperazine amides as novel c-jun N-terminal kinase (JNK) inhibitors.BDB
The Scripps Research Institute