15 articles for E Freire
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
Cmpds
Data
Article Title
Organization
22
Synthesis and cholinesterase inhibition of cativic acid derivatives.
Universidad Nacional Del Sur
12
Optimization of plasmepsin inhibitor by focusing on similar structural feature with chloroquine to avoid drug-resistant mechanism of Plasmodium falciparum.
Kyoto Pharmaceutical University
13
Synthesis and biochemical evaluation of triazole/tetrazole-containing sulfonamides against thrombin and related serine proteases.
The Johns Hopkins University
140
Design, synthesis and biological evaluation of small molecule inhibitors of CD4-gp120 binding based on virtual screening.
Bryn Mawr College
13
Improvement of both plasmepsin inhibitory activity and antimalarial activity by 2-aminoethylamino substitution.
Kyoto Pharmaceutical University
34
Antimalarial activity enhancement in hydroxymethylcarbonyl (HMC) isostere-based dipeptidomimetics targeting malarial aspartic protease plasmepsin.
Kyoto Pharmaceutical University
17
Additional interaction of allophenylnorstatine-containing tripeptidomimetics with malarial aspartic protease plasmepsin II.
Kyoto Pharmaceutical University
56
Synthetic, structural mimetics of the β-hairpin flap of HIV-1 protease inhibit enzyme function.
University of Maryland
15
New developments for the design, synthesis and biological evaluation of potent SARS-CoV 3CL(pro) inhibitors.
Kyoto Pharmaceutical University
16
A general strategy for creating "inactive-conformation" abl inhibitors.
The Scripps Research Institute