22 articles for A Christopoulos
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
Data
Article Title
Organization
Proof of concept study for designed multiple ligands targeting the dopamine D2, serotonin 5-HT2A, and muscarinic M1 acetylcholine receptors.
Monash University (Parkville Campus)
Molecular Mechanism of Action of Triazolobenzodiazepinone Agonists of the Type 1 Cholecystokinin Receptor. Possible Cooperativity across the Receptor Homodimeric Complex.
Mayo Clinic
Discovery, synthesis, and molecular pharmacology of selective positive allosteric modulators of thed-opioid receptor.
Bristol-Myers Squibb
Structure-activity relationships of privileged structures lead to the discovery of novel biased ligands at the dopamine D2 receptor.
Monash University
Synthesis and pharmacological evaluation of analogues of benzyl quinolone carboxylic acid (BQCA) designed to bind irreversibly to an allosteric site of the M1 muscarinic acetylcholine receptor.
Monash University (Parkville Campus)
A structure-activity analysis of biased agonism at the dopamine D2 receptor.
Monash University (Parkville Campus)
Allosteric modulation of seven transmembrane spanning receptors: theory, practice, and opportunities for central nervous system drug discovery.
Vanderbilt University Medical Center
Synthesis and SAR study of 4-arylpiperidines and 4-aryl-1,2,3,6-tetrahydropyridines as 5-HT2C agonists.
Monash University (Parkville Campus)
Discovery of antiandrogen activity of nonsteroidal scaffolds of marketed drugs.
The Scripps Research Institute
3- and 6-Substituted 2-amino-4,5,6,7-tetrahydrothieno[2,3-c]pyridines as A1 adenosine receptor allosteric modulators and antagonists.
Monash University (Parkville Campus)
2-aminothienopyridazines as novel adenosine A1 receptor allosteric modulators and antagonists.
Monash University
Synthesis and cannabinoid activity of 1-substituted-indole-3-oxadiazole derivatives: novel agonists for the CB1 receptor.
Monash University (Parkville Campus)
Structure-based virtual screening discovers potent and selective adenosine A
Uppsala University
The Design, Synthesis, and Evaluation of Novel 9-Arylxanthenedione-Based Allosteric Modulators for the δ
Monash University (Parkville Campus)
Probing structural requirements of positive allosteric modulators of the M4 muscarinic receptor.
Monash University
Synthesis and pharmacological profiling of analogues of benzyl quinolone carboxylic acid (BQCA) as allosteric modulators of the M1 muscarinic receptor.
Monash University
Synthesis and Pharmacological Evaluation of Heterocyclic Carboxamides: Positive Allosteric Modulators of the M
Monash University (Parkville Campus)
