23 articles for FX Tavares
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
Data
Article Title
Organization
The discovery and optimization of pyrimidinone-containing MCH R1 antagonists.
Glaxosmithkline
Anthranilimide-based glycogen phosphorylase inhibitors for the treatment of Type 2 diabetes: 2. Optimization of serine and threonine ether amino acid residues.
Glaxosmithkline
Anthranilimide-based glycogen phosphorylase inhibitors for the treatment of type 2 diabetes: 1. Identification of 1-amino-1-cycloalkyl carboxylic acid headgroups.
Glaxosmithkline
6-(4-chlorophenyl)-3-substituted-thieno[3,2-d]pyrimidin-4(3H)-one-based melanin-concentrating hormone receptor 1 antagonist.
Glaxosmithkline
Potent, selective, and orally efficacious antagonists of melanin-concentrating hormone receptor 1.
Glaxosmithkline
Ketoheterocycle-based inhibitors of cathepsin K: a novel entry into the synthesis of peptidic ketoheterocycles.
Glaxosmithkline
P2-P3 conformationally constrained ketoamide-based inhibitors of cathepsin K.
Glaxosmithkline
Ketoamide-based inhibitors of cysteine protease, cathepsin K: P3 modifications.
Glaxosmithkline
Potent and selective ketoamide-based inhibitors of cysteine protease, cathepsin K.
Glaxosmithkline
Orally bioavailable small molecule ketoamide-based inhibitors of cathepsin K.
Glaxosmithkline
Design of potent, selective, and orally bioavailable inhibitors of cysteine protease cathepsin k.
Glaxosmithkline
Small molecule DCN1 inhibitors and therapeutic methods using the same
University of Michigan
Amide compounds for treatment of immune and inflammatory disorders
Achillion Pharmaceuticals
Tricyclic fused pyridin-2-one derivatives and their use as BRD4 inhibitors
Jubilant Biosys
Pyrazolo-pyrrolidin-4-one derivatives as bet inhibitors and their use in the treatment of disease
Novartis
Bicyclic heteroaryl derivatives as CFTR potentiators
Cystic Fibrosis Foundation Therapeutics
S-imino-S-oxo-iminothiadiazine compounds as BACE inhibitors, compositions, and their use
Merck Sharp & Dohme
Dibenzofuran derivatives as inhibitors of fructose 1,6-bisphosphatase and methods of use thereof
Boston College
Detecting a quasi-stable imine species on the reaction pathway of SHV-1 ß-lactamase and 6ß-(hydroxymethyl)penicillanic acid sulfone.
Case Western Reserve University
17-hydroxy-19-nor-21-carboxylic acid-steroid γ-lactone derivative, use thereof, and medicament containing the derivative
TBA