17 articles for L Scapozza
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
Cmpds
Data
Article Title
Organization
3
Synthesis of 3-azabicyclo[3.2.2]nonanes and their antiprotozoal activities.

Karl-Franzens-University
3
Differences in conformational dynamics between Plasmodium falciparum and human Hsp90 orthologues enable the structure-based discovery of pathogen-selective inhibitors.

University of Geneva
16
Synthesis and biological evaluation of benzo[4,5]imidazo[1,2-c]pyrimidine and benzo[4,5]imidazo[1,2-a]pyrazine derivatives as anaplastic lymphoma kinase inhibitors.

University of Lyon
2
Synthesis and in vitro evaluation of a novel radioligand foravß3 integrin receptor imaging: [18F]FPPA-c(RGDfK).

University Hospital of Geneva
10
Design, synthesis, and biological and crystallographic evaluation of novel inhibitors of Plasmodium falciparum enoyl-ACP-reductase (PfFabI).

University of Bologna
38
Synthesis, structure-activity relationship and crystallographic studies of 3-substituted indolin-2-one RET inhibitors.

University of Milano-Bicocca
22
Inhibition of Plasmodium falciparum fatty acid biosynthesis: evaluation of FabG, FabZ, and FabI as drug targets for flavonoids.

University of Zurich
5
Development of a three-dimensional model for the N-methyl-D-aspartate NR2A subunit.

University of Milan
9
Synthesis and biological evaluation of 5-substituted derivatives of the potent antiherpes agent (north)-methanocarbathymine.

National Cancer Institute-Frederick
1
Discovery of the First Efficacious Adenosine 2A Receptor Negative Allosteric Modulators for High Adenosine Cancer Immunotherapies.

University of Geneva
3
Structural insights into the ATP binding pocket of the anaplastic lymphoma kinase by site-directed mutagenesis, inhibitor binding analysis, and homology modeling.

University of Milano-Bicocca
13
Identification of Natural Products Inhibiting SARS-CoV-2 by Targeting Viral Proteases: A Combined in Silico and in Vitro Approach.

University of Vienna
71
Identification of non-ATP-competitive α-carboline inhibitors of the anaplastic lymphoma kinase.

University of Milano-Bicocca
14
Ligand selectivity for the acetylcholine binding site of the rat alpha4beta2 and alpha3beta4 nicotinic subtypes investigated by molecular docking.

Swiss Federal Institute of Technology Zurich
19
Azetidine derivatives

Vernalis (R&D)
32
Cyclohexyl isoquinolinone compounds

Novartis
6
1,3-Di(2-[5-3H]tolyl)guanidine: a selective ligand that labels sigma-type receptors for psychotomimetic opiates and antipsychotic drugs.

The Oregon Health Sciences University