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16 articles for K Nakayama


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Identification of Novel D-Aspartate Oxidase Inhibitors by in Silico Screening and Their Functional and Structural Characterization in Vitro.EBI
Kitasato University
Discovery of novel 2-(alkylmorpholin-4-yl)-6-(3-fluoropyridin-4-yl)-pyrimidin-4(3H)-ones as orally-active GSK-3ß inhibitors for Alzheimer's disease.EBI
Mitsubishi Tanabe Pharma
Novel Indole-N-glucoside, TA-1887 As a Sodium Glucose Cotransporter 2 Inhibitor for Treatment of Type 2 Diabetes.EBI
Mitsubishi Tanabe Pharma
C-Glucosides with heteroaryl thiophene as novel sodium-dependent glucose cotransporter 2 inhibitors.EBI
Mitsubishi Tanabe Pharma
Discovery of canagliflozin, a novel C-glucoside with thiophene ring, as sodium-dependent glucose cotransporter 2 inhibitor for the treatment of type 2 diabetes mellitus.EBI
Mitsubishi Tanabe Pharma
Optimization of Novel Pyrido-pyridazinone Derivatives as FER Tyrosine Kinase Inhibitors, Leading to the Potent DS08701581.EBI
Daiichi Sankyo Co., Ltd.
MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 2: achieving activity in vivo through the use of alternative scaffolds.EBI
Daiichi Pharmaceutical
Structure-Based Design and Synthesis of an Isozyme-Selective MTHFD2 Inhibitor with a Tricyclic Coumarin Scaffold.EBI
Daiichi Sankyo
Discovery of a Potent, Selective, and Orally Available MTHFD2 Inhibitor (DS18561882) with in Vivo Antitumor Activity.EBI
Daiichi Sankyo
Discovery of Novel Pyrido-pyridazinone Derivatives as FER Tyrosine Kinase Inhibitors with Antitumor Activity.EBI
Daiichi Sankyo
Discovery of novel 2-(4-aryl-2-methylpiperazin-1-yl)-pyrimidin-4-ones as glycogen synthase kinase-3β inhibitors.EBI
Mitsubishi Tanabe Pharma
Synthesis, biochemical evaluation, and molecular modeling studies of aryl and arylalkyl di-n-butyl phosphates, effective butyrylcholinesterase inhibitors.EBI
California State University
Compounds useful for inhibiting RORγtBDB
Eli Lilly
Pyrazolopyridine derivative having GLP-1 receptor agonist effectBDB
Chugai Seiyaku Kabushiki Kaisha
A fragment-based approach to probing adenosine recognition sites by using dynamic combinatorial chemistry.BDB
University of Cambridge
2-Chloro-N6-cyclopentyladenosine: a highly selective agonist at A1 adenosine receptors.BDB
Pharmakologisches Institut, Heidelberg