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12 articles for C Valant


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Synthesis and pharmacological evaluation of analogues of benzyl quinolone carboxylic acid (BQCA) designed to bind irreversibly to an allosteric site of the M1 muscarinic acetylcholine receptor.EBI
Monash University (Parkville Campus)
Fluorescent derivatives of AC-42 to probe bitopic orthosteric/allosteric binding mechanisms on muscarinic M1 receptors.EBI
University of Strasburg
Synthesis and SAR study of 4-arylpiperidines and 4-aryl-1,2,3,6-tetrahydropyridines as 5-HT2C agonists.EBI
Monash University (Parkville Campus)
Allosteric functional switch of neurokinin A-mediated signaling at the neurokinin NK2 receptor: structural exploration.EBI
Umr Uds/Cnrs 7200
3- and 6-Substituted 2-amino-4,5,6,7-tetrahydrothieno[2,3-c]pyridines as A1 adenosine receptor allosteric modulators and antagonists.EBI
Monash University (Parkville Campus)
2-aminothienopyridazines as novel adenosine A1 receptor allosteric modulators and antagonists.EBI
Monash University
The Design, Synthesis, and Evaluation of Novel 9-Arylxanthenedione-Based Allosteric Modulators for the δEBI
Monash University (Parkville Campus)
Probing structural requirements of positive allosteric modulators of the M4 muscarinic receptor.EBI
Monash University
Synthesis and pharmacological profiling of analogues of benzyl quinolone carboxylic acid (BQCA) as allosteric modulators of the M1 muscarinic receptor.EBI
Monash University
Synthesis and Pharmacological Evaluation of Heterocyclic Carboxamides: Positive Allosteric Modulators of the MEBI
Monash University (Parkville Campus)
A Structure-Activity Relationship Study of Bitopic NEBI
Monash University
Structure-Based Design and Discovery of New MEBI
University of California