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28 articles for KT Lee


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
3,4-Dihydroquinazoline derivatives inhibit the activities of cholinesterase enzymes.EBI
Kyung Hee University
Synthesis, structure determination, and biological evaluation of phenylsulfonyl hydrazide derivatives as potential anti-inflammatory agents.EBI
Kyung Hee University
Hit-to-lead optimization of phenylsulfonyl hydrazides for a potent suppressor of PGE2 production: Synthesis, biological activity, and molecular docking study.EBI
Kyung Hee University
Discovery of 2-aryloxy-4-amino-quinazoline derivatives as novel protease-activated receptor 2 (PAR2) antagonists.EBI
Yonsei University
Targeting EGFR/HER2 tyrosine kinases with a new potent series of 6-substituted 4-anilinoquinazoline hybrids: Design, synthesis, kinase assay, cell-based assay, and molecular docking.EBI
Korea University of Science and Technology (Ust)
Computer-aided discovery of aminopyridines as novel JAK2 inhibitors.EBI
Chonnam National University
Synthesis and PGE2 production inhibition of s-triazine derivatives as a novel scaffold in RAW 264.7 macrophage cells.EBI
TBA
Inhibition of cellular proliferation and induction of apoptosis in human lung adenocarcinoma A549 cells by T-type calcium channel antagonist.EBI
Kyung Hee University
Synthesis, biological evaluation, and docking analysis of a novel family of 1-methyl-1H-pyrrole-2,5-diones as highly potent and selective cyclooxygenase-2 (COX-2) inhibitors.EBI
Kyung Hee University
Fragment-based discovery of novel and selective mPGES-1 inhibitors Part 1: identification of sulfonamido-1,2,3-triazole-4,5-dicarboxylic acid.EBI
Kyung Hee University
Identification of novel mPGES-1 inhibitors through screening of a chemical library.EBI
Kookmin University
Synthesis and antihypertensive activity of pyrimidin-4(3H)-one derivatives as losartan analogue for new angiotensin II receptor type 1 (AT1) antagonists.EBI
Kyung Hee University
In vivo evaluation of oral anti-tumoral effect of 3,4-dihydroquinazoline derivative on solid tumor.EBI
Kyung Hee University
Synthesis and PGE(2) production inhibition of 1H-furan-2,5-dione and 1H-pyrrole-2,5-dione derivatives.EBI
Kyung Hee University
Discovery of N-benzylbenzamide-based allosteric inhibitors of Aurora kinase A.EBI
Korea Institute of Science and Technology (KIST)
In vitro and in vivo neuroprotective effect of novel mPGES-1 inhibitor in animal model of Parkinson's disease.EBI
Kyung Hee University
Discovery of New Imidazo[2,1-EBI
National Research Centre (Nrc)
Optimization and Evaluation of Novel Antifungal Agents for the Treatment of Fungal Infection.EBI
Korea Institute of Science & Technology (Kist)
Discovery of N-amido-phenylsulfonamide derivatives as novel microsomal prostaglandin EEBI
Kyung Hee University
Design, synthesis, biological evaluation, and docking studies of novel (imidazol-5-yl)pyrimidine-based derivatives as dual BRAFEBI
Korea Institute of Science & Technology (Kist)
In vitro synergistic anticancer activity of the combination of T-type calcium channel blocker and chemotherapeutic agent in A549 cells.EBI
Kyung Hee University
Design, synthesis and anti-inflammatory activity of imidazol-5-yl pyridine derivatives as p38α/MAPK14 inhibitor.EBI
University of Science & Technology (Ust)
Thiazolidine-2,4-dione-based irreversible allosteric IKK-β kinase inhibitors: Optimization into in vivo active anti-inflammatory agents.EBI
Korea Institute of Science & Technology (Kist)
Synthesis and cytotoxic effects of 2-thio-3,4-dihydroquinazoline derivatives as novel T-type calcium channel blockers.EBI
Kyung Hee University
In vitro cytotoxicity on human ovarian cancer cells by T-type calcium channel blockers.EBI
Kyung Hee University
Design, synthesis and biological evaluation of novel thiazolidinedione derivatives as irreversible allosteric IKK-β modulators.EBI
Korea Institute of Science & Technology (Kist)
Novel LCK/FMS inhibitors based on phenoxypyrimidine scaffold as potential treatment for inflammatory disorders.EBI
Korea Institute of Science & Technology (Kist)
Synthesis and biological evaluation of fluoro-substituted 3,4-dihydroquinazoline derivatives for cytotoxic and analgesic effects.EBI
Kyung Hee University