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11 articles for thisTarget

The following articles (labelled with PubMed ID or TBD) are for your review

Article Title
Synthesis and biological evaluation of [125I]- and [123I]-4-iododexetimide, a potent muscarinic cholinergic receptor antagonist.EBI
Johns Hopkins Medical Institutions
Irreversible blockage of opioid receptor types by ester homologues of beta-funaltrexamine.EBI
Synthesis and biological activity of analogues of beta-chlornaltrexamine and beta-funaltrexamine at opioid receptors.EBI
Replacement of the peptide-backbone amides connecting Tyr-Gly and Gly-Gly in leucine-enkephalin with ketomethylene groups: synthesis and biological activity.EBI
Diastereomeric 6-desoxy-6-spiro-alpha-methylene-gamma-butyrolactone derivatives of naltrexone and oxymorphone. Selective irreversible inhibition of naltrexone binding in an opioid receptor preparation by a conformationally restricted michael acceptor ligand.EBI
N-Methylnalorphine: definition of N-allyl conformation for antagonism at the opiate receptor.EBI
Synthesis and pharmacology of metabolically stable tert-butyl ethers of morphine and levorphanol.EBI
Enkephalin glycopeptide analogues produce analgesia with reduced dependence liability.EBI
University of Northern Colorado
Opioid agonist and antagonist activities of morphindoles related to naltrindole.EBI
University of Minnesota
Structure-affinity relationship studies on 5-HT1A receptor ligands. 1. Heterobicyclic phenylpiperazines with N4-alkyl substituents.EBI
Solvay Duphar Research Laboratories
Design and synthesis of highly potent and selective cyclic dynorphin A analogues.EBI
University of Arizona