The first public molecular recognition database, BindingDB supports research, education and practice in drug discovery, pharmacology and related fields.

BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.6M data for 745K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

If BindingDB was of value to your research, please take a moment to donate to this nonprofit project. Your donation will let us provide you with more data and improved service.

To help with training and testing AI and other models, BindingDB downloads and search results now provide the publication date and BindingDB curation date of each measurement.

17 articles for G Ronsisvalle


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Multitarget opioid ligands in pain relief: New players in an old game.EBI
University of Catania
Evaluation of N-substitution in 6,7-benzomorphan compounds.EBI
University of Catania
Synthesis and structure-activity relationships of 1-aralkyl-4-benzylpiperidine and 1-aralkyl-4-benzylpiperazine derivatives as potent sigma ligands.EBI
University of Modena and Reggio Emilia
Synthesis of (+)-cis-N-(4-isothiocyanatobenzyl)-N-normetazocine, an isothiocyanate derivative of N-benzylnormetazocine as acylant agent for the sigma(1) receptor.EBI
University of Catania
Nonpeptide analogues of dynorphin A(1-8): design, synthesis, and pharmacological evaluation of kappa-selective agonists.EBI
University of Catania
Modeling of kappa-opioid receptor/agonists interactions using pharmacophore-based and docking simulations.EBI
University of Naples Federico II
(+)-cis-N-ethyleneamino-N-normetazocine derivatives. Novel and selective sigma ligands with antagonist properties.EBI
University of Catania
Non-peptide ligands for opioid receptors. Design of kappa-specific agonists.EBI
University of Catania
Hybrid bivalent ligands with opiate and enkephalin pharmacophores.EBI
University of Minnesota
Novel potent and selectives ligands: evaluation of their agonist and antagonist properties.EBI
University of Catania
Antiproliferative activity of phenylbutyrate ester of haloperidol metabolite II [(±)-MRJF4] in prostate cancer cells.EBI
University of Catania
Synthesis and resolution of cis-(+/-)-methyl (1R,2S/1S,2R)-2-[(4-hydroxy-4-phenylpiperidin-1-yl)methyl]-1-(4-methylphenyl)cyclopropanecarboxylate [(+/-)-PPCC)]: new sigma receptor ligands with neuroprotective effect.EBI
University of Catania
Novel sigma receptor ligands: synthesis and biological profile.EBI
University of Catania
Design, synthesis, and SAR analysis of novel selective sigma1 ligands.EBI
Università
6-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid mimics active conformation of tyrosine in opioid peptides.EBI
University of Catania
Kappa-opioid receptor model in a phospholipid bilayer: molecular dynamics simulation.EBI
University of Catania
Opioid agonist and antagonist bivalent ligands. The relationship between spacer length and selectivity at multiple opioid receptors.EBI
TBA