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17 articles for L Piemontese


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Cmpds
Data
Article Title
Organization
7
New diphenylmethane derivatives as peroxisome proliferator-activated receptor alpha/gamma dual agonists endowed with anti-proliferative effects and mitochondrial activity.EBI
University of Bari Aldo Moro
18
Design, synthesis and biological evaluation of a class of bioisosteric oximes of the novel dual peroxisome proliferator-activated receptora/ ligand LT175.EBI
University of Bari Aldo Moro
22
New 2-(aryloxy)-3-phenylpropanoic acids as peroxisome proliferator-activated receptora/¿ dual agonists able to upregulate mitochondrial carnitine shuttle system gene expression.EBI
Universit�
11
Synthesis, characterization and biological evaluation of ureidofibrate-like derivatives endowed with peroxisome proliferator-activated receptor activity.EBI
Istituto Tumori&Quot;Giovanni Paolo Ii&Quot
21
Synthesis, biological evaluation and molecular investigation of fluorinated peroxisome proliferator-activated receptorsa/¿ dual agonists.EBI
University of Bari Aldo Moro
20
New 2-aryloxy-3-phenyl-propanoic acids as peroxisome proliferator-activated receptors alpha/gamma dual agonists with improved potency and reduced adverse effects on skeletal muscle function.EBI
University of Bari Aldo Moro
24
Synthesis, biological evaluation, and molecular modeling investigation of chiral 2-(4-chloro-phenoxy)-3-phenyl-propanoic acid derivatives with PPARalpha and PPARgamma agonist activity.EBI
Università
9
A new potent and selective peroxisome proliferator-activated receptor alpha partial agonist displays anti-steatotic effects In vitro and behaves as a safe hypolipidemic and hypoglycemic agent in a diabetic mouse model.EBI
University of Bari
16
A chemical modification of a peroxisome proliferator-activated receptor pan agonist produced a shift to a new dual alpha/gamma partial agonist endowed with mitochondrial pyruvate carrier inhibition and antidiabetic properties.EBI
Universita degli Studi di Bari "Aldo Moro"
23
Chiral pyrrolidines as multipotent agents in Alzheimer and neurodegenerative diseases.EBI
Universita degli Studi di Bari
22
A chemoinformatics search for peroxisome proliferator-activated receptors ligands revealed a new pan-agonist able to reduce lipid accumulation and improve insulin sensitivity.EBI
Universit£?Degli Studi Di Bari "Aldo Moro
22
Structure-based design of novel donepezil-like hybrids for a multi-target approach to the therapy of Alzheimer's disease.EBI
University of Bari Aldo Moro
44
Virtual screening identification and chemical optimization of substituted 2-arylbenzimidazoles as new non-zinc-binding MMP-2 inhibitors.EBI
"A. Moro" University of Bari
7
An update about the crucial role of stereochemistry on the effects of Peroxisome Proliferator-Activated Receptor ligands.EBI
University of Bari Aldo Moro
3
New Approaches to Cancer Therapy: Combining Fatty Acid Amide Hydrolase (FAAH) Inhibition with Peroxisome Proliferator-Activated Receptors (PPARs) Activation.EBI
University of Bari Aldo Moro
24
Molecular determinants for nuclear receptors selectivity: chemometric analysis, dockings and site-directed mutagenesis of dual peroxisome proliferator-activated receptors α/γ agonists.EBI
University of Bari Aldo Moro
9
Identification of the First PPARα/γ Dual Agonist Able To Bind to Canonical and Alternative Sites of PPARγ and To Inhibit Its Cdk5-Mediated Phosphorylation.EBI
University of Bari Aldo Moro