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13 articles for MF Rafferty


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Synthesis, configuration, and evaluation of two conformationally restrained analogues of phencyclidine.EBI
National Institute of Diabetes, Digestive and Kidney Diseases
(S)-4-Methyl-2-(methylamino)pentanoic acid [4, 4-bis(4-fluorophenyl)butyl]amide hydrochloride, a novel calcium channel antagonist, is efficacious in several animal models of pain.EBI
Pfizer
Probes of the active site of norepinephrine N-methyltransferase: effect of hydrophobic and hydrophilic interactions on side-chain binding of amphetamine and alpha-methylbenzylamine.EBI
TBA
The design and synthesis of human branched-chain amino acid aminotransferase inhibitors for treatment of neurodegenerative diseases.EBI
Pfizer
Synthesis of a series of 4-benzyloxyaniline analogues as neuronal N-type calcium channel blockers with improved anticonvulsant and analgesic properties.EBI
Warner-Lambert
Structure-activity relationship at the proximal phenyl group in a series of non-peptidyl N-type calcium channel antagonists.EBI
Parke-Davis Pharmaceutical Research
Structure-activity relationship of N-methyl-N-aralkyl-peptidylamines as novel N-type calcium channel blockers.EBI
Warner-Lambert
Multiple parallel synthesis of N,N-dialkyldipeptidylamines as N-type calcium channel blockers.EBI
Warner-Lambert
Synthesis and biological evaluation of substituted 4-(OBz)phenylalanine derivatives as novel N-type calcium channel blockers.EBI
Warner-Lambert
N,N-dialkyl-dipeptidylamines as novel N-type calcium channel blockers.EBI
Warner-Lambert
Importance of the aromatic ring in adrenergic amines. 8. 2-(Aminomethyl)-trans-2-decalols as inhibitors of norepinephrine N-methyltransferase.EBI
TBA
Directional probes of the hydrophobic component of the aromatic ring binding site of norepinephrine N-methyltransferase.EBI
TBA
Importance of the aromatic ring in adrenergic amines. 7. Comparison of the stereoselectivity of norepinephrine N-methyltransferase for aromatic vs. nonaromatic substrates and inhibitors.EBI
TBA