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17 articles for I Enyedy


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of biaryl carboxylamides as potent ROR¿ inverse agonists.EBI
Biogen Idec
Discovery of novel pyrazole-containing benzamides as potent ROR¿ inverse agonists.EBI
Biogen
Structure-based design of low-nanomolar PIM kinase inhibitors.EBI
Biogen Idec
Synthesis and biological evaluation of 1-azabicyclo-[3.2.1]octanes: new dopamine transporter inhibitors.EBI
Georgetown University Medical Center
Identification and biochemical characterization of small-molecule inhibitors of Clostridium botulinum neurotoxin serotype A.EBI
U.S. Army Medical Research Institute of Infectious Diseases
3,5-diarylazoles as novel and selective inhibitors of protein kinase D.EBI
Novartis Institutes For Biomedical Research
Identification of potent and selective amidobipyridyl inhibitors of protein kinase D.EBI
Novartis Institutes For Biomedical Research
Identification of orally available naphthyridine protein kinase D inhibitors.EBI
Novartis Institutes For Biomedical Research
SAR of a novel 'Anthranilamide Like' series of VEGFR-2, multi protein kinase inhibitors for the treatment of cancer.EBI
Bayer Research Center
Substituted aminobenzimidazole pyrimidines as cyclin-dependent kinase inhibitors.EBI
Bayer Research Center
Discovery of Phospholipase D Inhibitors with Improved Drug-like Properties and Central Nervous System Penetrance.EBI
Biogen
Discovery of Potent, Selective, and Brain-Penetrant Apoptosis Signal-Regulating Kinase 1 (ASK1) Inhibitors that Modulate Brain Inflammation EBI
Biogen
Investigating small molecules to inhibit germinal center kinase-like kinase (GLK/MAP4K3) upstream of PKCθ phosphorylation: Potential therapy to modulate T cell dependent immunity.EBI
Biogen
Design, synthesis and identification of novel, orally bioavailable non-covalent Nrf2 activators.EBI
Biogen
Discovery of CNS-Penetrant Apoptosis Signal-Regulating Kinase 1 (ASK1) Inhibitors.EBI
Biogen
Rational Design and Optimization of a Novel Class of Macrocyclic Apoptosis Signal-Regulating Kinase 1 Inhibitors.EBI
TBA
Small molecules inhibit the interaction of Nrf2 and the Keap1 Kelch domain through a non-covalent mechanism.EBI
Biogen Idec