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20 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Cmpds
Data
Article Title
Organization
25
Pyrazoles as non-classical bioisosteres in prolylcarboxypeptidase (PrCP) inhibitors.EBI
Merck Research Laboratories
22
Discovery and optimization of orally active cyclohexane-based prolylcarboxypeptidase (PrCP) inhibitors.EBI
Merck Research Laboratories
23
A new class of prolylcarboxypeptidase inhibitors, part 2: the aminocyclopentanes.EBI
Merck Research Laboratories
37
A new class of prolylcarboxypeptidase inhibitors, part 1: discovery and evaluation.EBI
Merck Research Laboratories
43
Inhibitors of prolyl oligopeptidases for the therapy of human diseases: defining diseases and inhibitors.EBI
Mcgill University
10
Rigid phencyclidine analogues. Binding to the phencyclidine and sigma 1 receptors.EBI
University of Illinois At Chicago
39
Phencyclidine-like effects of tetrahydroisoquinolines and related compounds.EBI
G. D. Searle
38
Discovery of aminoheterocycles as potent and brain penetrant prolylcarboxypeptidase inhibitors.EBI
Merck Research Laboratories
24
Discovery of benzodihydroisofurans as novel, potent, bioavailable and brain-penetrant prolylcarboxypeptidase inhibitors.EBI
Merck Research Laboratories
26
Discovery of a new class of potent prolylcarboxypeptidase inhibitors derived from alanine.EBI
Merck Research Laboratories
46
The discovery of non-benzimidazole and brain-penetrant prolylcarboxypeptidase inhibitors.EBI
Merck Research Laboratories
33
Discovery of benzimidazole pyrrolidinyl amides as prolylcarboxypeptidase inhibitors.EBI
Merck Research Laboratories
62
Design and synthesis of prolylcarboxypeptidase (PrCP) inhibitors to validate PrCP as a potential target for obesity.EBI
Merck Research Laboratories
11
1'-Benzyl-3,4-dihydrospiro[2H-1- benzothiopyran-2,4'-piperidine] (spipethiane), a potent and highly selective sigma1 ligand.EBI
University of Camerino
11
Prolylcarboxypeptidase inhibitorsBDB
Merck Sharp & Dohme
32
Selective inhibitors of prolylcarboxypeptidaseBDB
University of Mississippi
10
Prolylcarboxypeptidase inhibitorsBDB
Merck Sharp & Dohme
9
Spiropiperidine prolylcarboxypeptidase inhibitorsBDB
Merck Sharp & Dohme
14
Prolylcarboxypeptidase inhibitorsBDB
Merck Sharp & Dohme
10
Prolylcarboxypeptidase inhibitorsBDB
Merck Sharp & Dohme