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9 articles for D Feytens


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Azepinone-Containing Tetrapeptide Analogues of Melanotropin Lead to Selective hMC4R Agonists and hMC5R Antagonist.EBI
Vrije Universiteit Brussel
Development and pharmacological characterization of conformationally constrained urotensin II-related peptide agonists.EBI
Laval University
The replacement of His(4) in angiotensin IV by conformationally constrained residues provides highly potent and selective analogues.EBI
Vrije Universiteit Brussel
Highly potent 4-amino-indolo[2,3-c]azepin-3-one-containing somatostatin mimetics with a range of sst receptor selectivities.EBI
Vrije Universiteit Brussel
Endomorphin-2 with a beta-turn backbone constraint retains the potent micro-opioid receptor agonist properties.EBI
Biological Research Center of The Hungarian Academy of Sciences
Design of novel neurokinin 1 receptor antagonists based on conformationally constrained aromatic amino acids and discovery of a potent chimeric opioid agonist-neurokinin 1 receptor antagonist.EBI
Vrije Universiteit Brussel
Novel multiple opioid ligands based on 4-aminobenzazepinone (Aba), azepinoindole (Aia) and tetrahydroisoquinoline (Tic) scaffolds.EBI
Vrije Universiteit Brussel
Conformationally constrained opioid ligands: the Dmt-Aba and Dmt-Aia versus Dmt-Tic scaffold.EBI
Vrije Universiteit Brussel
New sst4/5-selective somatostatin peptidomimetics based on a constrained tryptophan scaffold.EBI
Vrije Universiteit Brussel