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21 articles for M Koppitz


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Novel Mps1 Kinase Inhibitors with Potent Antitumor Activity.EBI
Bayer Pharma AG
Treating Cancer by Spindle Assembly Checkpoint Abrogation: Discovery of Two Clinical Candidates, BAY 1161909 and BAY 1217389, Targeting MPS1 Kinase.EBI
Bayer
Damage Incorporated: Discovery of the Potent, Highly Selective, Orally Available ATR Inhibitor BAY 1895344 with Favorable Pharmacokinetic Properties and Promising Efficacy in Monotherapy and in Combination Treatments in Preclinical Tumor Models.EBI
Bayer
Discovery and optimization of pyridyl-cycloalkyl-carboxylic acids as inhibitors of microsomal prostaglandin E synthase-1 for the treatment of endometriosis.EBI
Bayer
Discovery of BAY-298 and BAY-899: Tetrahydro-1,6-naphthyridine-Based, Potent, and Selective Antagonists of the Luteinizing Hormone Receptor Which Reduce Sex Hormone Levels in Vivo.EBI
Bayer
Crystalline succinate salt of 6-(6-aminopyrazin-2-yl)-n-(4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)imidazo[1,2-a]pyrazin-8-amineBDB
Kronos Bio
Inhibitors of tryptophan dioxygenases (IDO1 and TDO) and their use in therapyBDB
Auckland Uniservices
Substituted [5,6]cyclic-4(3H)-pyrimidinones as anticancer agentsBDB
Zenji Research Laboratories
PD-1/PD-L1 inhibitorsBDB
Gilead Sciences
Imidazolepyridine compounds and uses thereofBDB
Novartis
GLS1 inhibitors for treating diseaseBDB
The University of Texas System
Dihydroxy aromatic heterocyclic compoundBDB
Takeda Pharmaceutical
Molecular docking studies and biological evaluation of 1,3,4-thiadiazole derivatives bearing Schiff base moieties as tyrosinase inhibitors.BDB
Shaoyang University
Fused heterocyclic derivative, medicinal composition containing the same, and medicinal use thereofBDB
Kissei Pharmaceutical
Design, synthesis, biological evaluation, and molecular docking of novel benzopyran and phenylpyrazole derivatives as Akt inhibitors.BDB
Zhejiang University
Heterocyclic compounds and uses thereofBDB
Celgene Avilomics Research
Bicyclic compounds and their uses as dual c-SRC/JAK inhibitorsBDB
Debiopharm
Histone deacetylase inhibitors, process for preparation and uses thereofBDB
Zhejiang Hisun Pharmaceutical
Macrocyclic inhibitors of hepatitis C virusBDB
Medivir
Urokinase inhibitors, production and use thereofBDB
The Medicines