PMID
Data
Article Title
Organization
5-HT7 receptor modulators: Amino groups attached to biphenyl scaffold determine functional activity.

Yonsei University
Novel JAK1-selective benzimidazole inhibitors with enhanced membrane permeability.

Konkuk University
Novel N-acyl-carbazole derivatives as 5-HT7R antagonists.

Yonsei University
Benzimidazole Derivatives as Potent JAK1-Selective Inhibitors.

Konkuk University
Novel N-biphenyl-2-ylmethyl 2-methoxyphenylpiperazinylalkanamides as 5-HT7R antagonists for the treatment of depression.

Yonsei University
Novel thienopyrimidinones as mGluR1 antagonists.

Yonsei University
Discovery of aryl-biphenyl-2-ylmethylpiperazines as novel scaffolds for 5-HT(7) ligands and role of the aromatic substituents in binding to the target receptor.

Institute of Science and Technology
Synthesis and antibacterial activities of new piperidine substituted (5R)-[1,2,3]triazolylmethyl and (5R)-[(4-F-[1,2,3]triazolyl)methyl] oxazolidinones.

Korea Institute Science and Technology
Synthesis and biological evaluation of oxazole derivatives as T-type calcium channel blockers.

Institute of Science and Technology
Quinazolindione derivatives as potent 5-HT3A receptor antagonists.

Konkuk University
Novel quinazolinone derivatives as 5-HT7 receptor ligands.

Institute of Science and Technology
Novel GSK-3beta inhibitors from sequential virtual screening.

Korea Institute of Science and Technology
Design, synthesis, and biological evaluation of 1,3-dioxoisoindoline-5-carboxamide derivatives as T-type calcium channel blockers.

Institute of Science and Technology
The role of 2',3'-unsaturation on the antiviral activity of anti-HIV nucleosides against 3TC-resistant mutant (M184V).

The University of Georgia
Discovery of piperidinyl aminopyrimidine derivatives as IKK-2 inhibitors.

Korea Institute of Science and Technology
IKKbeta inhibitors identification part II: ligand and structure-based virtual screening.

Institute of Science and Technology
Identification of novel serotonin 2C receptor ligands by sequential virtual screening.

Institute of Science and Technology
IKKbeta inhibitors identification part I: homology model assisted structure based virtual screening.

Institute of Science and Technology
Discovery of novel amidobenzimidazole derivatives as orally available small molecule modulators of stimulator of interferon genes for cancer immunotherapy.

Korea Research Institute of Chemical Technology
Identification of (-)-Epigallocateshin gallate derivatives promoting innate immune activation via 2',3'-cyclic GMP-AMP-stimulator of interferon genes pathway.

Korea Institute of Science and Technology
3D pharmacophore based virtual screening of T-type calcium channel blockers.

Institute of Science and Technology
Novel T-type calcium channel blockers: dioxoquinazoline carboxamide derivatives.

Institute of Science and Technology
Discovery of G Protein-Biased Ligands against 5-HT

Korea Institute of Science and Technology
Discovery of G Protein-Biased Antagonists against 5-HT

Korea Institute of Science and Technology
Effects of fluorine substitution of cytosine analogues on the binding affinity to HIV-1 reverse transcriptase.

The University of Georgia
Synthesis and biological evaluation of picolinamides and thiazole-2-carboxamides as mGluR5 (metabotropic glutamate receptor 5) antagonists.

Korea Institute of Science & Technology (Kist)
Oxazolopyridines and thiazolopyridines as monoamine oxidase B inhibitors for the treatment of Parkinson's disease.

Korea Institute of Science and Technology
Synthesis and the 5-HT6 receptor antagonistic effect of 3-arylsulfonylamino-5,6-dihydro-6-substituted pyrazolo[3,4]pyridinones for neuropathic pain treatment.

Korea Institute of Science & Technology (Kist)
Discovery of β-Arrestin Biased Ligands of 5-HT

Korea Institute of Science and Technology
Neuropathic pain-alleviating effects of pyrazole-conjugated arylsulfonamides as 5-HT

University of Science and Technology
Phenyl-3,4-dihydroisoquinolin-2(1h)-yl-ethan-1-one derivatives as dopamine d1receptor positive allosteric modulators

Eli Lilly
Aminopyridazinone compounds as protein kinase inhibitors

Jiangsu Hengrui Medicine
4-substituted-cyclohexylamino-4-piperidinyl-acetamide antagonists of CCR2

Janssen Pharmaceutica
Evaluation of Coumarin and Neoflavone Derivatives as HCV NS5B Polymerase Inhibitors.

Umdnj-New Jersey Medical School