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15 articles for D Guiadeen


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Cmpds
Data
Article Title
Organization
30
Discovery of novel BTK inhibitors with carboxylic acids.EBI
Merck
6
Discovery of a Potent and Selective DGAT1 Inhibitor with a Piperidinyl-oxy-cyclohexanecarboxylic Acid Moiety.EBI
Merck Research Laboratories
21
Potent DGAT1 Inhibitors in the Benzimidazole Class with a Pyridyl-oxy-cyclohexanecarboxylic Acid Moiety.EBI
Merck Research Laboratories
100
1,3,8-Triazaspiro[4.5]decane-2,4-diones as efficacious pan-inhibitors of hypoxia-inducible factor prolyl hydroxylase 1-3 (HIF PHD1-3) for the treatment of anemia.EBI
Merck Research Laboratories
22
The synthesis and SAR of rhodanines as novel class C beta-lactamase inhibitors.EBI
The R. W. Johnson Pharmaceutical Research Institute
32
4-Amino-2-alkyl-butyramides as small molecule CCR2 antagonists with favorable pharmacokinetic properties.EBI
Merck Research Laboratories
27
Potent, non-covalent reversible BTK inhibitors with 8-amino-imidazo[1,5-a]pyrazine core featuring 3-position bicyclic ring substitutes.EBI
Merck
38
Discovery of 8-Amino-imidazo[1,5-a]pyrazines as Reversible BTK Inhibitors for the Treatment of Rheumatoid Arthritis.EBI
Merck Research Laboratories
22
Cholesteryl ester transfer protein (CETP) inhibitors based on cyclic urea, bicyclic urea and bicyclic sulfamide cores.EBI
Merck
13
Design, synthesis, and biological activity of diiminoisoindolines as complement component 3a antagonists.EBI
The R. W. Johnson Pharmaceutical Research Institute
53
Accelerating the discovery of DGAT1 inhibitors through the application of parallel medicinal chemistry (PMC).EBI
Merck
6
Benzimidazole-based DGAT1 inhibitors with a [3.1.0] bicyclohexane carboxylic acid moiety.EBI
Merck
23
Discovery of 3-morpholino-imidazole[1,5-a]pyrazine BTK inhibitors for rheumatoid arthritis.EBI
Merck
39
Benzodioxole derivative and preparation method and use thereofBDB
Zhejiang Hisun Pharmaceutical
50
Diamino heterocyclic carboxamide compoundBDB
Astellas Pharma