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14 articles for WG Humphreys


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Characterization of the in vitro and in vivo metabolism and disposition and cytochrome P450 inhibition/induction profile of saxagliptin in human.EBI
Bristol-Myers Squibb Research
Metabolic chiral inversion of brivanib and its relevance to safety and pharmacology.EBI
Bristol-Myers Squibb
(D)-2-tert-Butoxycarbonylamino-5,5-difluoro-5-phenyl-pentanoic acid: synthesis and incorporation into the growth hormone secretagogues.EBI
Bristol Myers Squibb
Comparative metabolism of radiolabeled muraglitazar in animals and humans by quantitative and qualitative metabolite profiling.EBI
Bristol-Myers Squibb
Optimization of 1H-tetrazole-1-alkanenitriles as potent orally bioavailable growth hormone secretagogues.EBI
Bristol-Myers Squibb Pharmaceutical Research Institute
Design and synthesis of tetrazole-based growth hormone secretagogue: the SAR studies of the O-benzyl serine side chain.EBI
Bristol Myers Squibb
Biphenylsulfonamide endothelin receptor antagonists. 4. Discovery of N-[[2'-[[(4,5-dimethyl-3-isoxazolyl)amino]sulfonyl]-4-(2-oxazolyl)[1,1'-biphenyl]- 2-yl]methyl]-N,3,3-trimethylbutanamide (BMS-207940), a highly potent and orally active ET(A) selective antagonist.EBI
Bristol-Myers Squibb Pharmaceutical Research Institute
Aglycone exploration of C-arylglucoside inhibitors of renal sodium-dependent glucose transporter SGLT2.EBI
Bristol Myers Squibb
Design and synthesis of N-[(4-methoxyphenoxy)carbonyl]-N-[[4-[2-(5- methyl-2-phenyl-4-oxazolyl)ethoxy]phenyl]methyl]glycine [Muraglitazar/BMS-298585], a novel peroxisome proliferator-activated receptor alpha/gamma dual agonist with efficacious glucose and lipid-lowering activities.EBI
Bristol-Myers Squibb Pharmaceutical Research Institute
6,7-dihydropyrido[2,1-A]phthalazin-2-ones for the treatment and prophylaxis of hepatitis B virus infectionBDB
Hoffmann-La Roche
Autotaxin inhibitorsBDB
Cancer Research Technology
Bicyclic heterocycles as FGFR4 inhibitorsBDB
Incyte
Substituted pyrido[3,4-b]pyrazines as GPR6 modulatorsBDB
Takeda Pharmaceutical
Pyridine derivatives as soft rock inhibitorsBDB
Redx Pharma