BDBM148430 US9682965, Compound A

SMILES [#6]-[#8]-[#6@@H]-1-[#6@@H](-[#6]-[#6][C@]2([#6]-[#8]2)[#6@H]-1[C@@]1([#6])[#8]-[#6@@H]1-[#6]\[#6]=[#6](\[#6])-[#6])-[#8]-[#6](=O)\[#6]=[#6]\c1ccc(-[#8]-[#6]-[#6]-[#7](-[#6])-[#6])cc1

InChI Key InChIKey=ZEZFKUBILQRZCK-MJSCXXSSSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 148430   

TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Zafgen

US Patent
LigandPNGBDBM148430(US9682965, Compound A)
Affinity DataIC50:  275nMpH: 7.4Assay Description:Flag tagged Human recombinant MetAP2 expressed and isolated for use as the enzyme source. 10 mM stock solutions of compounds were prepared in 100% DM...More data for this Ligand-Target Pair
In DepthDetails US Patent