BDBM24189 3-aminopropylphosphinic derivative, (R)-4::3-aminopropylphosphinic derivative, (S)-4::CGP44532::CHEMBL113304::CHEMBL113310::[(2S)-3-amino-2-hydroxypropyl](methyl)phosphinic acid
SMILES CP(O)(O)CC(=O)CN
InChI Key InChIKey=CLKFCXCQRLVUJX-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 24189
TargetGamma-aminobutyric acid (GABA) B receptor 1/type B receptor subunit 2 [41-940](Rat)
Astrazeneca
Astrazeneca
Affinity DataKi: 180nM ΔG°: -9.10kcal/mole EC50: 150nMpH: 7.4 T: 22°CAssay Description:Inhibition of [3H]GABA binding at GABAB receptor sites in rat brain synaptic membranes by test compounds was measured using a filtration binding assa...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid (GABA) B receptor 1/type B receptor subunit 2 [41-940](Rat)
Astrazeneca
Astrazeneca
Affinity DataKi: 840nM ΔG°: -8.20kcal/mole EC50: 600nMpH: 7.4 T: 22°CAssay Description:Inhibition of [3H]GABA binding at GABAB receptor sites in rat brain synaptic membranes by test compounds was measured using a filtration binding assa...More data for this Ligand-Target Pair