BDBM24189 3-aminopropylphosphinic derivative, (R)-4::3-aminopropylphosphinic derivative, (S)-4::CGP44532::CHEMBL113304::CHEMBL113310::[(2S)-3-amino-2-hydroxypropyl](methyl)phosphinic acid

SMILES CP(O)(O)CC(=O)CN

InChI Key InChIKey=CLKFCXCQRLVUJX-UHFFFAOYSA-N

Data  2 KI  6 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 24189   

TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM24189(3-aminopropylphosphinic derivative, (R)-4 | 3-amin...)
Affinity DataIC50:  5.40E+3nMAssay Description:Antagonist activity at human recombinant GABAc rho1 receptor expressed in Xenopus laevis oocytes at -60mV by two-electrode voltage clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM24189(3-aminopropylphosphinic derivative, (R)-4 | 3-amin...)
Affinity DataIC50:  1.71E+4nMAssay Description:Antagonist activity at human recombinant GABAc rho1 receptor expressed in Xenopus laevis oocytes at -60mV by two-electrode voltage clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed