BDBM284992 N-[2-fluoro-5-(2-methyl-1-oxoisoquinolin-4-yl) phenyl]methanesulfonamide::US10023592, Example 37
SMILES Cn1cc(-c2ccc(F)c(NS(C)(=O)=O)c2)c2ccccc2c1=O
InChI Key InChIKey=XAFXJYMUTUHGGU-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 284992
Affinity DataIC50: <500nMpH: 7.3Assay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair