BDBM285282 1,3-dimethyl-5-[3-methylsulfonyl-5-(pyridin-2- ylmethoxy)phenyl]pyridin-2-one::BDBM486126::US10023592, Example 330
SMILES Cc1cc(cn(C)c1=O)-c1cc(OCc2ccccn2)cc(c1)S(C)(=O)=O
InChI Key InChIKey=LRZHIMAYJUNZNR-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 285282
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair
Affinity DataIC50: <500nMpH: 7.3Assay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair