BDBM285441 N-[7-(1,5-dimethyl-6-oxopyridin-3-yl)-2- propyl-2,3-dihydro-1-benzofuran-5-yl] ethanesulfonamide::US10023592, Example 495::US10941160, Example 495
SMILES CCCC1Cc2cc(NS(=O)(=O)CC)cc(c2O1)-c1cc(C)c(=O)n(C)c1
InChI Key InChIKey=PBORVZVPTRTNPQ-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 285441
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair
Affinity DataIC50: <500nMpH: 7.3Assay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair