BDBM285454 5-(5-butyl-2-methylsulfonylpyrimidin-4-yl)-3- methyl-1-propan-2-ylpyridin-2-one::US10023592, Example 508::US10941160, Example 508
SMILES CCCCc1cnc(C)nc1-c1cc(C)c(=O)n(c1)C(C)C
InChI Key InChIKey=WQGAPIABMUQAJO-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 285454
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair
Affinity DataIC50: <500nMpH: 7.3Assay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair