BDBM285457 N-[5-butyl-4-(5-methyl-6-oxo-1-propan-2- ylpyridin-3-yl)pyrimidin-2-yl] ethanesulfonamide::US10023592, Example 511::US10941160, Example 511
SMILES CCCCc1cnc(CC)nc1-c1cc(C)c(=O)n(c1)C(C)C
InChI Key InChIKey=XLZQVAZBBXJXRD-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 285457
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair
Affinity DataIC50: <500nMpH: 7.3Assay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair