BDBM29094 (+/-)-SLV319::(S)-3-(4-chlorophenyl)-N-(4-chlorophenylsulfonyl)-N'-methyl-4-phenyl-4,5-dihydropyrazole-1-carboxamidine::3-(4-chlorophenyl)-N''''-(4-chlorophenylsulfonyl)-N-methyl-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamide::4-Chloro-N-[1-[3-(4-chloro-phenyl)-4-phenyl-4,5-dihydro-pyrazol-1-yl]-1-methylamino-meth-(E)-ylidene]-benzenesulfonamide::CHEMBL158784::SLV-319::ibipinabant
SMILES CN=C(NS(=O)(=O)c1ccc(Cl)cc1)N1CC(C(=N1)c1ccc(Cl)cc1)c1ccccc1
InChI Key InChIKey=AXJQVVLKUYCICH-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 29094
Affinity DataIC50: 139nMAssay Description:Inverse agonist activity against CB1 receptor expressed in human CHO cells assessed as effect on forskolin-stimulated cAMP levelMore data for this Ligand-Target Pair
Affinity DataIC50: 1.91nMAssay Description:Antagonist activity against human recombinant cannabinoid-1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Displacement of 3[H]ligand from recombinant human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+3nMAssay Description:Displacement of 3[H]ligand from recombinant human CB2 receptorMore data for this Ligand-Target Pair