BDBM35714 CHEMBL420762::Mozavaptan::N-[4-(5-Dimethylamino-2,3,4,5-tetrahydro-benzo[b]azepine-1-carbonyl)-phenyl]-2-methyl-benzamide::OPC-31260
SMILES CN(C)C1CCCN(C(=O)c2ccc(NC(=O)c3ccccc3C)cc2)c2ccccc12
InChI Key InChIKey=WRNXUQJJCIZICJ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 35714
TargetVasopressin V1a receptor(Human)
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
TargetVasopressin V1a receptor(Human)
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Affinity DataKi: 195nMAssay Description:Binding affinity to vasopressin V1a receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Displacement of [3H]-AVP from AVP-V1a receptor binding site in rat liverMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Human)
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Affinity DataIC50: 1.40E+3nMpH: 7.4 T: 4°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair