BDBM385795 3-(dimethylamino)propyl N- [5-(4-cyano-3-fluorophenyl)- [1,2,4]triazolo[1,5-a]pyridin- 7-yl]carbamate::US10287286, Example 198

SMILES CN(C)CCCOC(=O)Nc1cc(-c2ccc(C#N)c(F)c2)n2ncnc2c1

InChI Key InChIKey=GDKTZFXYPXBDTL-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 385795   

TargetProlyl hydroxylase EGLN2(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM385795(3-(dimethylamino)propyl N- [5-(4-cyano-3-fluorophe...)
Affinity DataIC50:  109nMAssay Description:The IC50 values for the PHD1 enzyme (residues 1-407) were determined by mixing increasing amounts of a compound of the invention with a fixed amount ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent