BDBM397088 4-Bromo-thiophene-2- carboxylic acid [4-(2- amino-ethoxy)-3-(4- chloro-2-methyl-2H- pyrazol-3-yl)-phenyl]- amide::US9987252, 77

SMILES Cn1ncc(Cl)c1-c1cc(NC(=O)c2cc(Br)cs2)ccc1OCCN


Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 397088   

Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM397088(4-Bromo-thiophene-2- carboxylic acid [4-(2- amino-...)
Affinity DataIC50:  1.20nMAssay Description:Radioligand binding assays for human 5-HT2A receptor was conducted using the 5-HT2 agonist [125I]DOI as radioligand. To define nonspecific binding, 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent