BDBM486259 3-(dimethylamino)-5-(2-ethoxy-5- ethylsulfonylphenyl)-1-methylpyridin-2-one::US10941160, Example 469
SMILES CCOc1ccc(cc1-c1cc(N(C)C)c(=O)n(C)c1)S(O)(O)CC
InChI Key InChIKey=TVVWMCXNTSIYMT-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 486259
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair