BDBM486274 N-[3-(1-cyclobutyl-5-methyl-6-oxopyridin-3- yl)-4-(2,4-difluorophenoxy)phenyl] methanesulfonamide::US10941160, Example 484
SMILES Cc1cc(cn(C2CCC2)c1=O)-c1cc(NS(C)=O)ccc1Oc1ccc(F)cc1F
InChI Key InChIKey=GFEYCDWOQUMYMW-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 486274
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair