BDBM486278 2-methyl-4-[5-(methylsulfonylmethyl)-2- (2,2,2-trifluoroethoxy)phenyl] isoquinolin-1-one::US10941160, Example 488
SMILES Cn1cc(-c2cc(CS(C)=O)ccc2OCC(F)(F)F)c2ccccc2c1=O
InChI Key InChIKey=GYFCYBBDMUOCQX-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 486278
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair