BDBM486280 N-[2-ethyl-8-(2-methyl-1-oxoisoquinolin-4-yl)- 3,4-difluoro-2H-chromen-6-yl] methanesulfonamide::US10941160, Example 490
SMILES CCC1CCc2cc(NS(C)=O)cc(c2O1)-c1cn(C)c(=O)c2ccccc12
InChI Key InChIKey=MXWBNPDWZMDJMC-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 486280
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair