BDBM50012956 1-cyclohexyl-3-(4-(2-(2-methylpyrazine-5-carboxamido)ethyl)phenylsulfonyl)urea::1-cyclohexyl-3-[[p-[2-(5-methylpyrazinecarboxamido)ethyl]phenyl]sulfonyl]urea::CHEMBL1073::CP-28720::GLIPIZIDE::Glucotrol::Glucotrol xl::K-4024::US20230348371, Compound Glipizide

SMILES Cc1cnc(cn1)C(=O)NCCc1ccc(cc1)S(=O)(=O)NC(=O)NC1CCCCC1

InChI Key InChIKey=ZJJXGWJIGJFDTL-UHFFFAOYSA-N

Data  7 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50012956   

TargetATP-binding cassette sub-family C member 4(Human)
Amgen

Curated by ChEMBL

LigandBDBM50012956(Glucotrol xl | Glucotrol | CHEMBL1073 | K-4024 | 1...)Copy SMILESCopy InChI

Affinity DataIC50: 1.33E+5nMAssay Description:Inhibition of human MRP4 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLDrugBankPC cidPC sidSimilars

In Depth
Date in BDB:
11/3/2019
Entry Details Article
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