BDBM50026614 CHEMBL575508
SMILES CC(C)[C@@H](CN1CC[C@](C)([C@@H](C)C1)c1cccc(O)c1)NC(=O)[C@H]1Cc2ccc(O)cc2CN1C
InChI Key InChIKey=OHIFKDNMHSXJFA-XAOJMSMDSA-N
Data 12 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 12 hits for monomerid = 50026614
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Science And Technology
Curated by ChEMBL
University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 0.0530nMAssay Description:Displacement of [3H]U69,593 from kappa opioid receptor in guinea pig brain membranes after 2 hrsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Science And Technology
Curated by ChEMBL
University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 0.0530nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
Affinity DataKi: 0.153nMAssay Description:Displacement of [3H]diprenorphine from human opioid kappa receptor expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity towards human cloned Opioid receptor kappa 1 using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Binding affinity towards human cloned Opioid receptor mu 1 using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Displacement of [3H]diprenorphine from human opioid mu receptor expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain tissueMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 118nMAssay Description:Binding affinity towards human cloned Opioid receptor delta 1 using [3H]Cl-DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: >500nMAssay Description:Displacement of [3H]diprenorphine from human opioid delta receptor expressed in HEK293 cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 616nMAssay Description:Inhibition of [3H]-DADLE binding to Opioid receptor delta 1 of rat brain tissueMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 616nMAssay Description:Displacement of [3H]DADLE from delta-opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair