BDBM50029644 CHEMBL296908::N-(3-(4-(4-(2-oxo-3,4-dihydroquinolin-1(2H)-yl)piperidine-1-carbonyl)phenoxy)propyl)acetamide::N-(3-{4-[4-(2-Oxo-3,4-dihydro-2H-quinolin-1-yl)-piperidine-1-carbonyl]-phenoxy}-propyl)-acetamide::OPC-1268::OPC-21268
SMILES CC(=O)NCCCOc1ccc(cc1)C(=O)N1CCC(CC1)N1C(=O)CCc2ccccc12
InChI Key InChIKey=KSNUCNRMDYJBKT-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 24 hits for monomerid = 50029644
Affinity DataKi: 23.5nMAssay Description:Binding affinity at Vasopressin V1a receptor, performed using [3H]-AVP on rat liverMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Evaluated for the binding affinity towards Vasopressin V1a receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity of the compound towards Vasopressin V1a receptor in rat liverMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity was evaluated by measuring the displacement of [3H]-AVP (arginine vasopressin) from specific binding sites in rat liver.More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Binding affinity was evaluated by measuring the displacement of [3H]-OT (oxytocin) from specific binding sites in uterine tissue obtained from human ...More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Binding affinity was evaluated by measuring the displacement of [3H]-OT (oxytocin) from specific binding sites in uterine tissue obtained from ratsMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Binding affinity to vasopressin V1a receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Evaluated for the binding affinity towards Vasopressin V2 receptor in rat kidney membrane using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity at cloned human Vasopressin V2 receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity at Vasopressin V2 receptor, performed using [3H]-AVP on rat kidneyMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Binding affinity of the compound towards Vasopressin V1a receptor in human liverMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+4nMAssay Description:Binding affinity was evaluated by measuring the displacement of [3H]-AVP (arginine vasopressin) from specific binding sites in kidney medulla obtaine...More data for this Ligand-Target Pair
Affinity DataKi: 5.20E+4nMAssay Description:Binding affinity was evaluated by measuring the displacement of [3H]-AVP (arginine vasopressin) from specific binding sites in human platelets.More data for this Ligand-Target Pair
Affinity DataKi: >8.10E+4nMAssay Description:Binding affinity was evaluated by measuring the displacement of [3H]-AVP (arginine vasopressin) from specific binding sites in kidney medulla obtaine...More data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Ability to displace [3H]- Arginine Vasopressin (AVP) from its specific binding sites in rat liver (V1 receptor)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Ability to displace [3H]- Arginine Vasopressin (AVP) from its specific binding sites in rat liver (V2 receptor)More data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Compound was evaluated for antagonistic activity against vasopressin V1 receptorMore data for this Ligand-Target Pair